化合物激酶活性测试-激酶抑制剂

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Kinase激酶
        酶学研究一直是药物研发的重要组成部分。合研生物拥有丰富的酶学筛选经验,酶学实验涵盖300多种筛选模型,包括了常见的组蛋白去乙酰酶类,组蛋白去甲基化酶,酪氨酸激酶,丝氨酸激酶,甲基化转移酶,磷酸二酯酶,DNA修复酶,热休克蛋白,免疫相关蛋白等。根据样本量的大小提供灵活的项目实施安排计划,可提供96孔和384孔两种板型的筛选模式,加速您的药物研发进程。

ABL1 ADP-Glo 96/384 well
ABL1(E255K) ADP-Glo 96/384 well
ABL1(T315I) ADP-Glo 96/384 well
ABL1(Y253F) ADP-Glo 96/384 well
ACK ADP-Glo 96/384 well
AKT1 ADP-Glo 96/384 well
AKT2 ADP-Glo 96/384 well
AKT3 ADP-Glo 96/384 well
ALK2 ADP-Glo 96/384 well
ALK4 ADP-Glo 96/384 well
ALK6 ADP-Glo 96/384 well
AMAPK(A1/B1/G2) ADP-Glo 96/384 well
AMPK(A1/B1/G1) ADP-Glo 96/384 well
AMPK(A2/B1/G1) ADP-Glo 96/384 well
ASK1 ADP-Glo 96/384 well
Aurora A ADP-Glo 96/384 well
Aurora B ADP-Glo 96/384 well
AXL ADP-Glo 96/384 well
BRK ADP-Glo 96/384 well
BXM ADP-Glo 96/384 well
CAMK1γ ADP-Glo 96/384 well
CAMK2α ADP-Glo 96/384 well
CAMK2γ ADP-Glo 96/384 well
CAMKK1 ADP-Glo 96/384 well
CDC7/DBF4 ADP-Glo 96/384 well
CDK2/CyclinA2 ADP-Glo 96/384 well
CDK2/CyclinE1 ADP-Glo 96/384 well
CDK3/cyclinE1 ADP-Glo 96/384 well
CDK5/p25 ADP-Glo 96/384 well
CDK5/p35 ADP-Glo 96/384 well
CDK6/CyclinD3 ADP-Glo 96/384 well
CDK9/Cyclink ADP-Glo 96/384 well
CHK1 ADP-Glo 96/384 well
CHK2 ADP-Glo 96/384 well
CK1a1 ADP-Glo 96/384 well
CK1γ1 ADP-Glo 96/384 well
CK1ε ADP-Glo 96/384 well
CK2α1 ADP-Glo 96/384 well
c-KIT ADP-Glo 96/384 well
CLK1 ADP-Glo 96/384 well
CLK3 ADP-Glo 96/384 well
c-MER ADP-Glo 96/384 well
CSK ADP-Glo 96/384 well
DAPK1 ADP-Glo 96/384 well
DDR2 ADP-Glo 96/384 well
DNA-PK ADP-Glo 96/384 well
DYRK2 ADP-Glo 96/384 well
EGFR ADP-Glo 96/384 well
EGFR(L858R) ADP-Glo 96/384 well
EGFR(L861Q) ADP-Glo 96/384 well
EGFR(T790,L858R) ADP-Glo 96/384 well
EGFR(T790M) ADP-Glo 96/384 well
EIF2AK2 ADP-Glo 96/384 well
EPHA1 ADP-Glo 96/384 well
ERK1 ADP-Glo 96/384 well
ERK2 ADP-Glo 96/384 well
FAK ADP-Glo 96/384 well
FES ADP-Glo 96/384 well
FGFR1 ADP-Glo 96/384 well
FGFR2 ADP-Glo 96/384 well
FGFR3(K650E) ADP-Glo 96/384 well
FGFR4 ADP-Glo 96/384 well
FLT1 ADP-Glo 96/384 well
FLT3 ADP-Glo 96/384 well
FLT3(D835Y) ADP-Glo 96/384 well
FMS ADP-Glo 96/384 well
FYN A ADP-Glo 96/384 well
GRK5 ADP-Glo 96/384 well
GSK3α ADP-Glo 96/384 well
GSK3β ADP-Glo 96/384 well
HER2 ADP-Glo 96/384 well
HER4 ADP-Glo 96/384 well
HIPK1 ADP-Glo 96/384 well
HPK1 ADP-Glo 96/384 well
IGF1R ADP-Glo 96/384 well
IKKß ADP-Glo 96/384 well
IKKα ADP-Glo 96/384 well
InsR ADP-Glo 96/384 well
IRAK4 ADP-Glo 96/384 well
ITK ADP-Glo 96/384 well
JAK3 ADP-Glo 96/384 well
JNK1 ADP-Glo 96/384 well
JNK3 ADP-Glo 96/384 well
KDR ADP-Glo 96/384 well
KHS1 ADP-Glo 96/384 well
LCK ADP-Glo 96/384 well
Lipid kinase ADP-Glo 96/384 well
LRRK2 ADP-Glo 96/384 well
LYN B ADP-Glo 96/384 well
MAPKAPK2 ADP-Glo 96/384 well
MAPKAPK3 ADP-Glo 96/384 well
MAPKAPK5 ADP-Glo 96/384 well
MARK1 ADP-Glo 96/384 well
MELK ADP-Glo 96/384 well
MET ADP-Glo 96/384 well
MET(M1250T) ADP-Glo 96/384 well
MINK1 ADP-Glo 96/384 well
MLCK ADP-Glo 96/384 well
MLK1 ADP-Glo 96/384 well
MLK2 ADP-Glo 96/384 well
MRCKa ADP-Glo 96/384 well
MSK1 ADP-Glo 96/384 well
MSK2 ADP-Glo 96/384 well
MST1 ADP-Glo 96/384 well
MYO3β ADP-Glo 96/384 well
Name ADP-Glo 96/384 well
NEK2 ADP-Glo 96/384 well
NEK3 ADP-Glo 96/384 well
NIK ADP-Glo 96/384 well
NUAK2 ADP-Glo 96/384 well
p38B ADP-Glo 96/384 well
p38α ADP-Glo 96/384 well
p38γ ADP-Glo 96/384 well
P38δ ADP-Glo 96/384 well
p70S6K ADP-Glo 96/384 well
p70S6Kb ADP-Glo 96/384 well
PAK1/CDC42 ADP-Glo 96/384 well
PAK3 ADP-Glo 96/384 well
PAK4 ADP-Glo 96/384 well
PASK ADP-Glo 96/384 well
PDGFRa(D842V) ADP-Glo 96/384 well
PDGFRa(T674I) ADP-Glo 96/384 well
PDGFRα ADP-Glo 96/384 well
PDGFRβ ADP-Glo 96/384 well
PDK1 ADP-Glo 96/384 well
PI3K Lipid kinases ADP-Glo 96/384 well
PI3K-Glo ADP-Glo 96/384 well
PIM1 ADP-Glo 96/384 well
PIM2 ADP-Glo 96/384 well
PKA ADP-Glo 96/384 well
PKC ADP-Glo 96/384 well
PKCß1 ADP-Glo 96/384 well
PKCα ADP-Glo 96/384 well
PKCβII ADP-Glo 96/384 well
PKCγ ADP-Glo 96/384 well
PKCδ ADP-Glo 96/384 well
PKCε ADP-Glo 96/384 well
PKCζ ADP-Glo 96/384 well
PKCθ ADP-Glo 96/384 well
PKCι ADP-Glo 96/384 well
PKCμ ADP-Glo 96/384 well
PKD2 ADP-Glo 96/384 well
PLK1 ADP-Glo 96/384 well
PRKG1 ADP-Glo 96/384 well
PYK2 ADP-Glo 96/384 well
RET ADP-Glo 96/384 well
RET(V804L) ADP-Glo 96/384 well
RET(Y791F) ADP-Glo 96/384 well
RIPK2 ADP-Glo 96/384 well
ROCK1 ADP-Glo 96/384 well
ROCK2 ADP-Glo 96/384 well
RON ADP-Glo 96/384 well
RSK1 ADP-Glo 96/384 well
SGK1 ADP-Glo 96/384 well
SIK ADP-Glo 96/384 well
SLK ADP-Glo 96/384 well
SRC ADP-Glo 96/384 well
STK33 ADP-Glo 96/384 well
SYK ADP-Glo 96/384 well
TAK1-TAB1 ADP-Glo 96/384 well
TAOK1 ADP-Glo 96/384 well
TBK1 ADP-Glo 96/384 well
TGFbR1 ADP-Glo 96/384 well
TGFβR2 ADP-Glo 96/384 well
TNIK ADP-Glo 96/384 well
TOPK ADP-Glo 96/384 well
TRKA ADP-Glo 96/384 well
TRKB ADP-Glo 96/384 well
ULK1 ADP-Glo 96/384 well
VRK2 ADP-Glo 96/384 well
WNK1 ADP-Glo 96/384 well
ZAK ADP-Glo 96/384 well
ZAP70 ADP-Glo 96/384 well