Kinase激酶
酶学研究一直是药物研发的重要组成部分。合研生物拥有丰富的酶学筛选经验,酶学实验涵盖300多种筛选模型,包括了常见的组蛋白去乙酰酶类,组蛋白去甲基化酶,酪氨酸激酶,丝氨酸激酶,甲基化转移酶,磷酸二酯酶,DNA修复酶,热休克蛋白,免疫相关蛋白等。根据样本量的大小提供灵活的项目实施安排计划,可提供96孔和384孔两种板型的筛选模式,加速您的药物研发进程。
ABL1 | ADP-Glo | 96/384 well |
ABL1(E255K) | ADP-Glo | 96/384 well |
ABL1(T315I) | ADP-Glo | 96/384 well |
ABL1(Y253F) | ADP-Glo | 96/384 well |
ACK | ADP-Glo | 96/384 well |
AKT1 | ADP-Glo | 96/384 well |
AKT2 | ADP-Glo | 96/384 well |
AKT3 | ADP-Glo | 96/384 well |
ALK2 | ADP-Glo | 96/384 well |
ALK4 | ADP-Glo | 96/384 well |
ALK6 | ADP-Glo | 96/384 well |
AMAPK(A1/B1/G2) | ADP-Glo | 96/384 well |
AMPK(A1/B1/G1) | ADP-Glo | 96/384 well |
AMPK(A2/B1/G1) | ADP-Glo | 96/384 well |
ASK1 | ADP-Glo | 96/384 well |
Aurora A | ADP-Glo | 96/384 well |
Aurora B | ADP-Glo | 96/384 well |
AXL | ADP-Glo | 96/384 well |
BRK | ADP-Glo | 96/384 well |
BXM | ADP-Glo | 96/384 well |
CAMK1γ | ADP-Glo | 96/384 well |
CAMK2α | ADP-Glo | 96/384 well |
CAMK2γ | ADP-Glo | 96/384 well |
CAMKK1 | ADP-Glo | 96/384 well |
CDC7/DBF4 | ADP-Glo | 96/384 well |
CDK2/CyclinA2 | ADP-Glo | 96/384 well |
CDK2/CyclinE1 | ADP-Glo | 96/384 well |
CDK3/cyclinE1 | ADP-Glo | 96/384 well |
CDK5/p25 | ADP-Glo | 96/384 well |
CDK5/p35 | ADP-Glo | 96/384 well |
CDK6/CyclinD3 | ADP-Glo | 96/384 well |
CDK9/Cyclink | ADP-Glo | 96/384 well |
CHK1 | ADP-Glo | 96/384 well |
CHK2 | ADP-Glo | 96/384 well |
CK1a1 | ADP-Glo | 96/384 well |
CK1γ1 | ADP-Glo | 96/384 well |
CK1ε | ADP-Glo | 96/384 well |
CK2α1 | ADP-Glo | 96/384 well |
c-KIT | ADP-Glo | 96/384 well |
CLK1 | ADP-Glo | 96/384 well |
CLK3 | ADP-Glo | 96/384 well |
c-MER | ADP-Glo | 96/384 well |
CSK | ADP-Glo | 96/384 well |
DAPK1 | ADP-Glo | 96/384 well |
DDR2 | ADP-Glo | 96/384 well |
DNA-PK | ADP-Glo | 96/384 well |
DYRK2 | ADP-Glo | 96/384 well |
EGFR | ADP-Glo | 96/384 well |
EGFR(L858R) | ADP-Glo | 96/384 well |
EGFR(L861Q) | ADP-Glo | 96/384 well |
EGFR(T790,L858R) | ADP-Glo | 96/384 well |
EGFR(T790M) | ADP-Glo | 96/384 well |
EIF2AK2 | ADP-Glo | 96/384 well |
EPHA1 | ADP-Glo | 96/384 well |
ERK1 | ADP-Glo | 96/384 well |
ERK2 | ADP-Glo | 96/384 well |
FAK | ADP-Glo | 96/384 well |
FES | ADP-Glo | 96/384 well |
FGFR1 | ADP-Glo | 96/384 well |
FGFR2 | ADP-Glo | 96/384 well |
FGFR3(K650E) | ADP-Glo | 96/384 well |
FGFR4 | ADP-Glo | 96/384 well |
FLT1 | ADP-Glo | 96/384 well |
FLT3 | ADP-Glo | 96/384 well |
FLT3(D835Y) | ADP-Glo | 96/384 well |
FMS | ADP-Glo | 96/384 well |
FYN A | ADP-Glo | 96/384 well |
GRK5 | ADP-Glo | 96/384 well |
GSK3α | ADP-Glo | 96/384 well |
GSK3β | ADP-Glo | 96/384 well |
HER2 | ADP-Glo | 96/384 well |
HER4 | ADP-Glo | 96/384 well |
HIPK1 | ADP-Glo | 96/384 well |
HPK1 | ADP-Glo | 96/384 well |
IGF1R | ADP-Glo | 96/384 well |
IKKß | ADP-Glo | 96/384 well |
IKKα | ADP-Glo | 96/384 well |
InsR | ADP-Glo | 96/384 well |
IRAK4 | ADP-Glo | 96/384 well |
ITK | ADP-Glo | 96/384 well |
JAK3 | ADP-Glo | 96/384 well |
JNK1 | ADP-Glo | 96/384 well |
JNK3 | ADP-Glo | 96/384 well |
KDR | ADP-Glo | 96/384 well |
KHS1 | ADP-Glo | 96/384 well |
LCK | ADP-Glo | 96/384 well |
Lipid kinase | ADP-Glo | 96/384 well |
LRRK2 | ADP-Glo | 96/384 well |
LYN B | ADP-Glo | 96/384 well |
MAPKAPK2 | ADP-Glo | 96/384 well |
MAPKAPK3 | ADP-Glo | 96/384 well |
MAPKAPK5 | ADP-Glo | 96/384 well |
MARK1 | ADP-Glo | 96/384 well |
MELK | ADP-Glo | 96/384 well |
MET | ADP-Glo | 96/384 well |
MET(M1250T) | ADP-Glo | 96/384 well |
MINK1 | ADP-Glo | 96/384 well |
MLCK | ADP-Glo | 96/384 well |
MLK1 | ADP-Glo | 96/384 well |
MLK2 | ADP-Glo | 96/384 well |
MRCKa | ADP-Glo | 96/384 well |
MSK1 | ADP-Glo | 96/384 well |
MSK2 | ADP-Glo | 96/384 well |
MST1 | ADP-Glo | 96/384 well |
MYO3β | ADP-Glo | 96/384 well |
Name | ADP-Glo | 96/384 well |
NEK2 | ADP-Glo | 96/384 well |
NEK3 | ADP-Glo | 96/384 well |
NIK | ADP-Glo | 96/384 well |
NUAK2 | ADP-Glo | 96/384 well |
p38B | ADP-Glo | 96/384 well |
p38α | ADP-Glo | 96/384 well |
p38γ | ADP-Glo | 96/384 well |
P38δ | ADP-Glo | 96/384 well |
p70S6K | ADP-Glo | 96/384 well |
p70S6Kb | ADP-Glo | 96/384 well |
PAK1/CDC42 | ADP-Glo | 96/384 well |
PAK3 | ADP-Glo | 96/384 well |
PAK4 | ADP-Glo | 96/384 well |
PASK | ADP-Glo | 96/384 well |
PDGFRa(D842V) | ADP-Glo | 96/384 well |
PDGFRa(T674I) | ADP-Glo | 96/384 well |
PDGFRα | ADP-Glo | 96/384 well |
PDGFRβ | ADP-Glo | 96/384 well |
PDK1 | ADP-Glo | 96/384 well |
PI3K Lipid kinases | ADP-Glo | 96/384 well |
PI3K-Glo | ADP-Glo | 96/384 well |
PIM1 | ADP-Glo | 96/384 well |
PIM2 | ADP-Glo | 96/384 well |
PKA | ADP-Glo | 96/384 well |
PKC | ADP-Glo | 96/384 well |
PKCß1 | ADP-Glo | 96/384 well |
PKCα | ADP-Glo | 96/384 well |
PKCβII | ADP-Glo | 96/384 well |
PKCγ | ADP-Glo | 96/384 well |
PKCδ | ADP-Glo | 96/384 well |
PKCε | ADP-Glo | 96/384 well |
PKCζ | ADP-Glo | 96/384 well |
PKCθ | ADP-Glo | 96/384 well |
PKCι | ADP-Glo | 96/384 well |
PKCμ | ADP-Glo | 96/384 well |
PKD2 | ADP-Glo | 96/384 well |
PLK1 | ADP-Glo | 96/384 well |
PRKG1 | ADP-Glo | 96/384 well |
PYK2 | ADP-Glo | 96/384 well |
RET | ADP-Glo | 96/384 well |
RET(V804L) | ADP-Glo | 96/384 well |
RET(Y791F) | ADP-Glo | 96/384 well |
RIPK2 | ADP-Glo | 96/384 well |
ROCK1 | ADP-Glo | 96/384 well |
ROCK2 | ADP-Glo | 96/384 well |
RON | ADP-Glo | 96/384 well |
RSK1 | ADP-Glo | 96/384 well |
SGK1 | ADP-Glo | 96/384 well |
SIK | ADP-Glo | 96/384 well |
SLK | ADP-Glo | 96/384 well |
SRC | ADP-Glo | 96/384 well |
STK33 | ADP-Glo | 96/384 well |
SYK | ADP-Glo | 96/384 well |
TAK1-TAB1 | ADP-Glo | 96/384 well |
TAOK1 | ADP-Glo | 96/384 well |
TBK1 | ADP-Glo | 96/384 well |
TGFbR1 | ADP-Glo | 96/384 well |
TGFβR2 | ADP-Glo | 96/384 well |
TNIK | ADP-Glo | 96/384 well |
TOPK | ADP-Glo | 96/384 well |
TRKA | ADP-Glo | 96/384 well |
TRKB | ADP-Glo | 96/384 well |
ULK1 | ADP-Glo | 96/384 well |
VRK2 | ADP-Glo | 96/384 well |
WNK1 | ADP-Glo | 96/384 well |
ZAK | ADP-Glo | 96/384 well |
ZAP70 | ADP-Glo | 96/384 well |