激酶(kinase)是最大且功能最多样的基因家族之一,同时也是重要的药物靶点。激酶是细胞功能的关键调节分子。合研生物提供多种类型激酶靶点,为激酶药物筛选提供基于生化检测及细胞检测服务,还可根据客户药物筛选需求提供多样性激酶谱服务。
Target | Assay | Format |
ABL1 | ADP-Glo | 96/384 well |
ABL1(E255K) | ADP-Glo | 96/384 well |
ABL1(T315I) | ADP-Glo | 96/384 well |
ABL1(Y253F) | ADP-Glo | 96/384 well |
ACK | ADP-Glo | 96/384 well |
AKT1 | ADP-Glo | 96/384 well |
AKT2 | ADP-Glo | 96/384 well |
AKT3 | ADP-Glo | 96/384 well |
ALK2 | ADP-Glo | 96/384 well |
ALK4 | ADP-Glo | 96/384 well |
ALK6 | ADP-Glo | 96/384 well |
AMAPK(A1/B1/G2) | ADP-Glo | 96/384 well |
AMPK(A1/B1/G1) | ADP-Glo | 96/384 well |
AMPK(A2/B1/G1) | ADP-Glo | 96/384 well |
ASK1 | ADP-Glo | 96/384 well |
Aurora A | ADP-Glo | 96/384 well |
Aurora B | ADP-Glo | 96/384 well |
AXL | ADP-Glo | 96/384 well |
BRK | ADP-Glo | 96/384 well |
BXM | ADP-Glo | 96/384 well |