合研生物拥有丰富的酶学筛选经验,酶学实验涵盖几百种筛选模型(其中激酶300多种),包括了常见的组蛋白去乙酰酶类,组蛋白去甲基化酶,酪氨酸激酶,丝氨酸激酶,甲基化转移酶,磷酸二酯酶,DNA修复酶,热休克蛋白,免疫相关蛋白等,根据样本量的大小提供灵活的项目实施安排计划,可提供96孔和384孔两种板型的筛选模式,加速您的药物研发进程。除针对激酶的测试外,其他酶学靶点的测试也是药物研发的重要组成部分。
Bromodomains
Target | Assay | Format |
ATAD2A | TR-FRET/AlphaScreen assay | 96/384 well |
ATAD2B | TR-FRET/AlphaScreen assay | 96/384 well |
BACE1 | TR-FRET | 96/384 well |
BAZ2B | AlphaScreen assay | 96/384 well |
BPTF/FALZ | TR-FRET | 96/384 well |
BRD1 | TR-FRET/AlphaScreen assay | 96/384 well |
BRD2 | TR-FRET/AlphaScreen assay | 96/384 well |
BRD3 | TR-FRET/AlphaScreen assay | 96/384 well |
BRD4 | TR-FRET/AlphaScreen assay | 96/384 well |
BRD9 | TR-FRET | 96/384 well |
BRDT | TR-FRET | 96/384 well |
BRG1 | TR-FRET | 96 well |
BRM | TR-FRET | 96 well |
BRPF3 | TR-FRET/AlphaScreen assay | 96/384 well |
CBP | TR-FRET | 96 well |
CECR2 | TR-FRET/AlphaScreen assay | 96/384 well |
CREBBP | TR-FRET/AlphaScreen assay | 96/384 well |
SMARCA2 | TR-FRET/AlphaScreen assay | 96/384 well |
SMARCA4 | TR-FRET/AlphaScreen assay | 96/384 well |
TAF1(BD2) | TR-FRET | 96/384 well |
TAF1L(BD2) | TR-FRET | 96/384 well |
TRIM24 | TR-FRET | 96/384 well |
WDR9/BRWD1 | TR-FRET | 96/384 well |