其他酶学功能检测

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        合研生物拥有丰富的酶学筛选经验,酶学实验涵盖几百种筛选模型(其中激酶300多种),包括了常见的组蛋白去乙酰酶类,组蛋白去甲基化酶,酪氨酸激酶,丝氨酸激酶,甲基化转移酶,磷酸二酯酶,DNA修复酶,热休克蛋白,免疫相关蛋白等,根据样本量的大小提供灵活的项目实施安排计划,可提供96孔和384孔两种板型的筛选模式,加速您的药物研发进程。除针对激酶的测试外,其他酶学靶点的测试也是药物研发的重要组成部分。

Bromodomains

Target Assay Format
ATAD2A TR-FRET/AlphaScreen assay 96/384 well
ATAD2B TR-FRET/AlphaScreen assay 96/384 well
BACE1 TR-FRET 96/384 well
BAZ2B AlphaScreen assay 96/384 well
BPTF/FALZ TR-FRET 96/384 well
BRD1 TR-FRET/AlphaScreen assay 96/384 well
BRD2 TR-FRET/AlphaScreen assay 96/384 well
BRD3 TR-FRET/AlphaScreen assay 96/384 well
BRD4 TR-FRET/AlphaScreen assay 96/384 well
BRD9 TR-FRET 96/384 well
BRDT TR-FRET 96/384 well
BRG1 TR-FRET 96 well
BRM TR-FRET 96 well
BRPF3 TR-FRET/AlphaScreen assay 96/384 well
CBP TR-FRET 96 well
CECR2 TR-FRET/AlphaScreen assay 96/384 well
CREBBP TR-FRET/AlphaScreen assay 96/384 well
SMARCA2 TR-FRET/AlphaScreen assay 96/384 well
SMARCA4 TR-FRET/AlphaScreen assay 96/384 well
TAF1(BD2) TR-FRET 96/384 well
TAF1L(BD2) TR-FRET 96/384 well
TRIM24 TR-FRET 96/384 well
WDR9/BRWD1 TR-FRET 96/384 well